An investigation of (R)-(+)-1-(1-naphthyl)ethylimines and (R)-(+)-1-(phenyl)ethylimines as chiral templates in the Staudinger reactionGEORG, G. I; ZHIJUN WU.Tetrahedron letters. 1994, Vol 35, Num 3, issn 0040-4039, 343, 381-384 [5 p.]Article

Stereoselective syn aldol raction of the lithium ester enolate of ethyl N,N-dimethylglycine in the presence of triethylboraneGEORG, G. I; AKGÜN, E.Tetrahedron letters. 1991, Vol 32, Num 40, pp 5521-5524, issn 0040-4039Article

An asymmetric synthesis of carbapenem antibiotic (+)-PS-5 from ethyl 3-hydroxybutanoateGEORG, G. I; KANT, J.Journal of organic chemistry. 1988, Vol 53, Num 3, pp 692-695, issn 0022-3263Article

Enantioselective synthesis of a 3'-dephenylcryptophycin synthonEGGEN, M; GEORG, G. I.Bioorganic & medicinal chemistry letters (Print). 1998, Vol 8, Num 22, pp 3177-3180, issn 0960-894XArticle

Metal directed stereoselective synthesis of 3-(1'-hydroxyethyl)-2-azetidinones from ethyl 3-hydroxybutyrateGEORG, G. I; AKGUÊN, E.Tetrahedron letters. 1990, Vol 31, Num 23, pp 3267-3270, issn 0040-4039, 4 p.Article

Internal nucleophile assisted selective deesterification studies on baccatin III. Synthesis of 2-debenzoyl- and 4-deacetylbaccatin III analoguesAPURBA DATTA; JAYASINGHE, L. R; GEORG, G. I et al.Journal of organic chemistry. 1994, Vol 59, Num 16, pp 4689-4690, issn 0022-3263Article

4-Deacetyltaxol and 10-acetyl-4-deacetyltaxotere : synthesis and biological evaluationAPURBA DATTA; JAYASINGHE, L. R; GEORG, G. I et al.Journal of medicinal chemistry (Print). 1994, Vol 37, Num 24, pp 4258-4260, issn 0022-2623Article

Substituted 6-alkyloxapenems: potent β-lactamase inhibitors; synthesis and biological characterizationWILD, H; METZGER, K.-G.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 11, pp 2205-2210, issn 0960-894XArticle

Asymmetric synthesis of (1'R,3R,4R)-4-acetoxy-3-1'-((tert-butyldimethylsilyl)oxy)ethyl-2-azetidinonnes and other 3-(1'hydroxyethyl)-2-azetidiones from (S)-(+)-ethyl 3-hydroxybutanoate: formal total synthesis of (+)-thienamycinGEORG, G. I; KANT, J; GILL, H. S et al.Journal of the American Chemical Society. 1987, Vol 109, Num 4, pp 1129-1135, issn 0002-7863Article

3-(1'-Hydroxyethyl)-2-azetidinones from 3-hydroxybutyrates and N-arylaldiminesGEORG, G. I; GILL, H. S; GERHARDT, C et al.Tetrahedron letters. 1985, Vol 26, Num 33, pp 3903-3906, issn 0040-4039Article

Stereo- and enantio-controlled synthesis of chiral intermediates for the total synthesis of thienamycin and related β-lactam antibiotics from 3-hydroxybutyratesGEORG, G. I; GILL, H. S.Journal of the Chemical Society. Chemical communications. 1985, Num 20, pp 1433-1435, issn 0022-4936Article

Rearrangement of unsymmetrical azetidinone disulfides to 2β-(heterocyclylthiomethyl)penams, a synthetic approach to new β-lactamase inhibitorsVON DAEHNE, W; HOFFMEYER, L; KEIDING, J et al.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 11, pp 2247-2252, issn 0960-894XArticle

Cyclopentenones as potential inhibitors of penicillin sensitive enzymesDURAND, T; MARCHAND-BRYNAERT, J; GHOSEZ, L et al.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 11, pp 2309-2312, issn 0960-894XArticle

Synthesis and biological activity of tetracyclic carbapenemsSCHMIDT, G; SCHRÖCK, W; ENDERMANN, R et al.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 11, pp 2193-2198, issn 0960-894XArticle

3-Phosphono-1-carba-1-dethiacephalosporins as antibacterial agentsTERNANSKY, R. J; PIKE, A. J.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 11, pp 2237-2240, issn 0960-894XArticle

Synthesis and antibacterial activity of (1'R,5R,6R)-2-tert-butyl-6-(1'-hydroxyethyl)oxapenem-3-carboxylic acidPFAENDLER, H. R; WEISNER, F; METZGER, K et al.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 11, pp 2211-2218, issn 0960-894XArticle

Halohydrin analogues of cryptophycin 1 : Synthesis and biological activityGEORG, G. I; ALI, S. M; STELLA, V. J et al.Bioorganic & medicinal chemistry letters (Print). 1998, Vol 8, Num 15, pp 1959-1962, issn 0960-894XArticle

Taxol photoaffinity labels. II: Synthesis and biological evaluation of N-(4-azidobenzoyl)-N-debenzoyltaxol, N-(4-azido-2,3,5,6-tetrafluorobenzoyl)-N-debenzoyltaxol, and 7-(4-azido-2,3,5,6-tetrafluorozoyl)taxolGEORG, G. I; HARRIMAN, G. C. B; HAEIL PARK et al.Bioorganic & medicinal chemistry letters (Print). 1994, Vol 4, Num 3, pp 487-490, issn 0960-894XArticle

The effect of the aromatic rings of taxol on biological activity and solution conformation : synthesis and evaluation of saturated taxol and taxotere analoguesBOGE, T. CH; HIMES, R. H; VANDER VELDE, D. G et al.Journal of medicinal chemistry (Print). 1994, Vol 37, Num 20, pp 3337-3343, issn 0022-2623Article

Activity of new penems against defined MRSA strainsJABES, D; ROSSI, R; DELLA BRUNA, C et al.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 11, pp 2165-2170, issn 0960-894XArticle

Taxol photoaffinity label: 7-(p-azidobenzoyl)taxol synthesis and biological evaluationGEORG, G. I; HARRIMAN, G. C. B; HIMES, R. H et al.Bioorganic & medicinal chemistry letters. 1992, Vol 2, Num 7, 640, 735-738 [5 p.]Article

A one-step synthesis of a deuterated paclitaxel analogue : 10-deacetoxy-(10α-²H)paclitaxelDUTTA, D; HADD, H; VANDER VELDE, D. G et al.Bioorganic & medicinal chemistry letters (Print). 1999, Vol 9, Num 23, pp 3277-3278, issn 0960-894XArticle

Heteroaromatic taxol analogues : the chemistry and biological activities of 3'-furyl and 3'-pyridyl substituted taxanesGEORG, G. I; HARRIMAN, G. C. B; HEPPERLE, M et al.Bioorganic & medicinal chemistry letters (Print). 1994, Vol 4, Num 11, pp 1381-1384, issn 0960-894XArticle

Structure-activity studies of antitumor taxanes : synthesis of novel C-13 side chain homologated taxol and taxotere analogsJAYASINGHE, L. R; DATTA, A; ALI, S. M et al.Journal of medicinal chemistry (Print). 1994, Vol 37, Num 18, pp 2981-2984, issn 0022-2623Article

Hydrophobic collapse of taxol and taxotere solution conformations in mixtures of water and organic solventVANDER VELDE, D. G; GEORG, G. I; GRUNEWALD, G. L et al.Journal of the American Chemical Society. 1993, Vol 115, Num 24, pp 11650-11651, issn 0002-7863Article